Rimegepant

Definition

Rimegepant is a calcitonin gene-related peptide (CGRP) receptor antagonist used for the acute treatment of migraine headaches. It works by blocking the CGRP receptors to alleviate migraine symptoms.

5 Must Know Facts For Your Next Test

1. Rimegepant is administered orally and is available in tablet form.
2. It provides relief from migraine pain within two hours of administration.
3. Rimegepant can be used with or without food, offering flexibility in dosing.
4. Common side effects include nausea and hypersensitivity reactions.
5. It should not be used concomitantly with strong CYP3A4 inhibitors or inducers.

Review Questions

• What class of drug is Rimegepant?
• How does Rimegepant alleviate migraine symptoms?
• Name two common side effects of Rimegepant.

Related terms

CGRP Receptor Antagonist: A class of drugs that block calcitonin gene-related peptide receptors to treat migraines.

Migraine Headache: A neurological condition characterized by intense, debilitating headaches often accompanied by nausea, vomiting, and sensitivity to light and sound.

CYP3A4 Inhibitors: Drugs that inhibit the enzyme CYP3A4, affecting the metabolism of various medications including rimegepant.